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東莞市景源實(shí)驗(yàn)科技有限公司
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硼替佐米雜質(zhì)有哪些

時(shí)間:2023/10/11閱讀:814
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東莞市景源實(shí)驗(yàn)科技有限公司可提供硼替佐米雜質(zhì)全套,并隨貨提供COA證書,HPLC,NMR,MS圖譜,10mg/25mg/50mg/100mg/500mg等多種規(guī)格可選,更大規(guī)格需確認(rèn)庫存。我司可根據(jù)客戶需要提供硼替佐米雜質(zhì)定制服務(wù)。


硼替佐米的相關(guān)介紹

硼替佐米(Bortezomib),為黃色固體的化學(xué)品,商品名 :萬珂® VELCADE®,中文別名:MG-341;硼替佐米雜質(zhì);保特佐米,熔點(diǎn):122-124°C,分子式 :C19H25BN4O4,分子量 :384.23700,用于既往未經(jīng)治療的且不適合大劑量化療和骨髓抑制的多發(fā)性骨髓瘤患者的治療;或單藥用于至少接受過一種或一種以上治療后復(fù)發(fā)的多發(fā)性骨髓瘤患者的治療;本品可用于復(fù)發(fā)或難治性套細(xì)胞淋巴瘤患者的治療,此患者在使用本品前至少接受過一種治療。用于該適應(yīng)癥的安全有效性數(shù)據(jù)來自國外一項(xiàng)針對(duì)既往治療后復(fù)發(fā)的套細(xì)胞淋巴瘤的單臂Ⅱ期臨床研究,尚缺乏針對(duì)中國人群的臨床研究數(shù)據(jù)。


硼替佐米雜質(zhì)有哪些


中文名稱

英文名稱

CAS號(hào)

硼替佐米標(biāo)準(zhǔn)品

Bortezomib

179324-69-7

硼替佐米雜質(zhì)1

Bortezomib Amide Analog

289472-80-6

硼替佐米雜質(zhì)2

Bortezomib Acid Analog

114457-94-2

硼替佐米雜質(zhì)3

Bortezomib (2R)-Acid

1608986-16-8

硼替佐米雜質(zhì)4

Desisobutyl-n-butyl Bortezomib

1104011-35-9

硼替佐米雜質(zhì)5

(1R, 2R)-Bortezomib

1132709-15-9

硼替佐米雜質(zhì)6

(1S, 2S)-Bortezomib

1132709-14-8

硼替佐米雜質(zhì)7

(1S, 2R)-Bortezomib

1132709-16-0

硼替佐米雜質(zhì)8

PS-619


硼替佐米雜質(zhì)9

Bortezomib Hydroxy (1R, 2S)-Isomer,(R)-Hydroxy Des(boric Acid) Bortezomib

289472-78-2

硼替佐米雜質(zhì)10

Bortezomib Hydroxy (1R, 2R)-Isomer,(R,R)-Hydroxy Des(boric Acid) Bortezomib


硼替佐米雜質(zhì)11

Bortezomib Hydroxy (1S, 2S)-Isomer,(R)-Hydroxy Des(boric Acid) Bortezomib

289472-81-7

硼替佐米雜質(zhì)12

Bortezomib Acid Methyl Ester

73058-37-4

硼替佐米雜質(zhì)13

Bortezomib Pinanediol Impurity,(1R)-(S)-Pinanediol-N-(2-pyrazinylcarbonyl)-L-phenylalanine-L-leucine boronate

205393-22-2

硼替佐米雜質(zhì)14

Bortezomib Impurity N,(R)-Hydroperoxy Des(boric Acid) Bortezomib,Bortezomib R-Hydroxyperoxide

886979-78-8

硼替佐米雜質(zhì)15

Bortezomib Impurity M,(S)-Hydroperoxy Des(boric Acid) Bortezomib,Bortezomib R-Hydroxyperoxide

886979-81-3

硼替佐米雜質(zhì)16

N-((S)-1-(((S)-1-methoxy-3-methylbutyl)amino)-1-oxo-3-phenylpropan-2-yl)pyrazine-2-carboxamide


硼替佐米雜質(zhì)17

N-((S)-1-(((S)-1-methoxy-3-methylbutyl)amino)-1-oxo-3-phenylpropan-2-yl)pyrazine-2-carboxamide


硼替佐米雜質(zhì)18

(S)-N-(1-(isopentylamino)-1-oxo-3-phenylpropan-2-yl)pyrazine-2-carboxamide

1446194-56-4

硼替佐米雜質(zhì)19

(S,E)-N-(1-((3-methylbut-1-en-1-yl)amino)-1-oxo-3-phenylpropan-2-yl)pyrazine-2-carboxamide


硼替佐米雜質(zhì)20

(S)-N-(1-formamido-1-oxo-3-phenylpropan-2-yl)pyrazine-2-carboxamide


硼替佐米雜質(zhì)21

3-Hydroxy Bortezomib


硼替佐米雜質(zhì)22

Bortezomib N-Hexyl Impurity,Desisobutyl-n-pentyl Bortezomib


硼替佐米雜質(zhì)23

Bortezomib L-Phenylalanyl Analog,L-Phenylalanine-bortezomib

1194235-41-0

硼替佐米雜質(zhì)24

Bortezomib D-Phenylalanyl Analog,D-Phenylalanine-bortezomib






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